Crisaborole
Ko Crisaborole he mema o te karaehe o te benzoxaboroles he 5-hydroxy-1,3-dihydro-2,1-benzoxaborole kei roto te phenolic.hauwaikua whakakapihia e te roopu 4-cyanophenyl. He aukati phosphodiesterase 4 e whakamahia ana mo te maimoatanga o te mate ngawari ki te ngawari o te mate o nga tamariki me nga pakeke. He mahi hei aukati phosphodiesterase IV, heantisoriaticme te tarukino anti-inflammatory kore-steroidal. He benzoxaborole, he ether kakara me te nitrile.
He pūrākau a Crisaboroleoxaborolei whakaaetia e te FDA i te Hakihea 14, 2016 hei Eucrisa, he maimoatanga mo te mate mo te ngawari me te ngawari o te mate pukupuku. Ko tenei kaihoko kore-steroidal he kaha ki te whakapai ake i te kaha o te mate, te whakaiti i te mate o te mate me te whakaiti i nga tohu me nga tohu i roto i nga turoro 2 tau me te pakeke ake. Ka whakaitihia te mumura o te rohe i roto i te kiri me te aukati i te kaha ake o te mate me te tohu haumaru pai. Kei roto i tona hanganga aboronngota, e whakahaere ana i te urunga o te kiri me te here ki te pokapū bimetal o te phosphodiesterase 4 enzyme. I tenei wa kei te whakawhanakehia hei maimoatanga kaupapa mo te psoriasis.
Ko te Crisaborole he Phosphodiesterase 4 Inhibitor. Ko te tikanga o te mahi o te crisaborole ko te Phosphodiesterase 4 Inhibitor.
Tono18Ko nga kaupapa Aromātai Tauritenga Kounga kua whakaaetia4, a6kei te whakamanahia nga kaupapa.
Ko te punaha whakahaere kounga teitei o te ao kua whakatakoto he turanga pakari mo nga hoko.
Ko te tirotiro i te kounga ka haere i roto i te huringa ora katoa o te hua ki te whakarite i te kounga me te hua rongoa.
Ko te roopu Whakahaere Whakahaere Ngaio e tautoko ana i nga tono kounga i te wa o te tono me te rehitatanga.
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